发明名称 INTERMEDIATES AND METHODS USEFUL IN THE SEMISYNTHESIS OF PACLITAXEL AND ANALOGS
摘要 The semisynthesis of paclitaxel and its analogs uses new intermediates which are derivatives of 10-deacetyl-baccatin III, the invention also provides methods for preparing these derivatives. These novel derivatives have alkyl carbonate or alkyl carbonyl substituents in the 7 position.
申请公布号 WO9926939(A1) 申请公布日期 1999.06.03
申请号 WO1998IB01912 申请日期 1998.11.19
申请人 INDENA S.P.A.;BOMBARDELLI, EZIO 发明人 BOMBARDELLI, EZIO
分类号 C07D305/14;A61K31/337;A61P35/00;C07D263/04;C07D263/06;C07F7/18;(IPC1-7):C07D305/14 主分类号 C07D305/14
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