发明名称 Synthesis of swainsonine salts
摘要 A method for synthesizing swainsonine salts and intermediates thereof comprising subjecting a compound of the formula I wherein R2 and R2' are the same or different and represent alkyl, halogen, alkenyl, alkoxy, cycloalkyl or aryl which may be substituted, to acid hydrolysis in the presence of a C1-4 alkanol to obtain a crystalline salt of swainsonine; and optionally, recrystallizing the swainsonine salt from a C1-4 alkanol. The reaction may be used in combination with one or more additional reaction steps.
申请公布号 AU9617298(A) 申请公布日期 1999.05.17
申请号 AU19980096172 申请日期 1998.10.23
申请人 GLYCODESIGN INC. 发明人 FRANCOIS TROPPER;RAJAN N. SHAH;PRADEEP SHARMA
分类号 A61K31/437;A61P43/00;C07D317/30;C07D471/04;C07D491/056;C07D491/14;C07D491/147;C07D491/18 主分类号 A61K31/437
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