发明名称 |
PROCESS OF CONVERTING TAXANES INTO BACCATIN III AND 10-DEACETYLBACCATIN III |
摘要 |
A process for the preparation of a compound of formula (II) where R1 = H or R1 = COCH3, comprising contacting a mixture containing at least one taxane compound having an ester linkage at the C -13 position with at least one borohydride reducing salt in a reaction solvent in the presence of a Lewis acid.
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申请公布号 |
CA2142354(C) |
申请公布日期 |
1999.05.04 |
申请号 |
CA19932142354 |
申请日期 |
1993.08.16 |
申请人 |
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发明人 |
CARVER, DAVID R.;PROUT, TIMOTHY R.;EWALD, HERNITA A.;HENDERSON, DONIA L. |
分类号 |
C07D305/14;(IPC1-7):C07D305/14 |
主分类号 |
C07D305/14 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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