发明名称 8-SUBSTITUTED-9H-1,3-DIOXOLO/4,5-h//2,3/BENZODIAZEPINE DERIVATIVES, AS AMPA/KAINATE RECEPTOR INHIBITORS
摘要 The invention refers to novel 8-substituted-9H-1,3-dioxolo/4,5-h//2,3/benzodiazepine derivatives of formula (I), a process for preparing these compounds and to pharmaceutical compositions containing these active substances. Compounds (I) inhibit Ampa/Kainate receptors.
申请公布号 WO9907707(A1) 申请公布日期 1999.02.18
申请号 WO1998HU00075 申请日期 1998.08.07
申请人 EGIS GYOGYSZERGYAR RT.;RATKAI, ZOLTAN;BARKOCZY, JOZSEF;SCHNEIDER, GEZA;CSELENYAK, JUDIT;SIMIG, GYULA;BALAZS, LASZLO;DOMAN, IMRE;GREFF, ZOLTAN;KOTAY NAGY, PETER;SERES, PETER;SZABO, GEZA;GACSALYI, ISTVAN;GIGLER, GABOR;GYERTYAN, ISTVAN;LEVAY, GYOERGY;KOVACS, ATTILA;SIMO, ANNAMARIA;SZABADOS, TAMAS;EGYED, ANDRAS;VEGH, MIKLOS;TIHANYI, KAROLY 发明人 RATKAI, ZOLTAN;BARKOCZY, JOZSEF;SCHNEIDER, GEZA;CSELENYAK, JUDIT;SIMIG, GYULA;BALAZS, LASZLO;DOMAN, IMRE;GREFF, ZOLTAN;KOTAY NAGY, PETER;SERES, PETER;SZABO, GEZA;GACSALYI, ISTVAN;GIGLER, GABOR;GYERTYAN, ISTVAN;LEVAY, GYOERGY;KOVACS, ATTILA;SIMO, ANNAMARIA;SZABADOS, TAMAS;EGYED, ANDRAS;VEGH, MIKLOS;TIHANYI, KAROLY
分类号 A61K31/551;A61P1/08;A61P21/02;A61P25/00;A61P25/06;A61P25/08;A61P25/28;C07D491/04;C07D491/056;(IPC1-7):C07D491/04;A61K31/55 主分类号 A61K31/551
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