发明名称 |
PHARMACEUTICAL COMPOSITIONS AND METHODS FOR EFFECTING DOPAMINE RELEASE |
摘要 |
Patients susceptible to or suffering from disorders, such as central nervous system disorders, which are characterized by an alteration in normal neurotransmitter release, such as dopamine release (e.g., Parkinsonism, Parkinson's Disease, Tourette's Syndrome, attention deficient disorder, or schizophrenia) are treated by administering an endo or exo form of a 1-aza-2-(3-pyridyl)bicyclo¢2.2.1!heptane, a 1-aza-2-(3-pyridyl)bicyclo¢2.2.2! octane, a 1-aza-2-(3-pyridyl)bicyclo¢3.2.2!nonane, a 1aza-7-(3-pyridyl) bicyclo¢2.2.1!heptane, a 1-aza-3-(3-pyridyl)bicyclo¢3.2.2!nonane, or a 1-aza-7-(3-pyridyl)bicyclo¢3.2.2!nonane.
|
申请公布号 |
CA2294990(A1) |
申请公布日期 |
1999.01.07 |
申请号 |
CA19982294990 |
申请日期 |
1998.04.22 |
申请人 |
UNIVERSITY OF KENTUCKY RESEARCH FOUNDATION;R.J. REYNOLDS TOBACCO COMPANY |
发明人 |
DULL, GARY MAURICE;BHATTI, BALWINDER SINGH;CALDWELL, WILLIAM SCOTT;LIPPIELLO, PATRICK MICHAEL;CROOKS, PETER ANTHONY;DEO, NIRANJAN MADHUKAR;BENCHERIF, MEROUANE;RAVARD, ALAIN |
分类号 |
A61K31/407;A61K31/439;A61K31/55;A61P25/00;A61P25/16;A61P25/28;C07D453/02;C07D471/08;C07D487/08;(IPC1-7):C07D453/02;A61K31/44 |
主分类号 |
A61K31/407 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|