发明名称 TRICYCLIC PYRROLE OR PYRAZOLE DERIVATIVE
摘要 Tricyclic pyrrole or pyrazole derivatives represented by general formula (I) or pharmaceutically acceptable salts thereof, which have high selectivity and affinity for 5-HT2c receptors and are useful in treating central nervous system diseases such as sexual function disorder, appetite regulation disorder, anxiety, depression or sleep disturbance. In said formula, the ring Y represents an unsaturated 5-membered ring optionally having 1 to 3 heteroatoms of one or more types selected from the group consisting of nitrogen, oxygen and sulfur or an unsaturated 6-membered ring having 1 or 2 nitrogen atoms; X represents a bond or carbon; --- represents a double or single bond; V represents nitrogen or CH; and A represents linear or branched lower alkylene optionally substituted by halogeno or cycloalkyl.
申请公布号 CA2291651(A1) 申请公布日期 1998.12.17
申请号 CA19982291651 申请日期 1998.06.11
申请人 YAMANOUCHI PHARMACEUTICAL CO., LTD. 发明人 SAKAMOTO, SHUICHI;KIMIZUKA, TETSUYA;SHIMADA, ITSURO;KUBOTA, HIDEKI;MAENO, KYOICHI;KAZUTA, KEN-ICHI;WANIBUCHI, FUMIKAZU
分类号 A61K31/381;A61K31/415;A61K31/4162;C07D231/54;C07D491/04;C07D491/048;C07D495/04;C07D498/04;C07D513/04;(IPC1-7):C07D231/54;C07D471/04;A61K31/40;A61K31/42;A61K31/425;A61K31/47;A61K31/55 主分类号 A61K31/381
代理机构 代理人
主权项
地址