发明名称 COUMARIN DERIVATIVES, METHODS OF PREPARATION AND APPLICATION AS MEDICINES
摘要 The invention concerns compounds of general formula (I) in which: X, X' and X'' independently of each other represent O or S; Y represents O, S, NH or NHS; R3 represents in particular a cycloalkyl group; R5, R6, R7 and R8 mutually identical or different, represent in particular hydrogen; a halogen atom. Said compounds can be used as active substances of medicines as inhibitors of protease.
申请公布号 WO9855472(A1) 申请公布日期 1998.12.10
申请号 WO1998FR01087 申请日期 1998.05.29
申请人 CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE;REBOUD-RAVAUX, MICHELE;POCHET, LIONEL;DOUCET, CAROLINE;PIROTTE, BERNARD;BOGGETTO, NICOLE;DELARGE, JACQUES 发明人 REBOUD-RAVAUX, MICHELE;POCHET, LIONEL;DOUCET, CAROLINE;PIROTTE, BERNARD;BOGGETTO, NICOLE;DELARGE, JACQUES
分类号 A61K31/37;A61K31/4433;A61K31/4436;A61K31/453;A61K31/4709;A61K31/4725;A61P1/18;A61P7/02;A61P9/10;A61P11/00;A61P13/12;A61P17/00;A61P19/02;A61P29/00;A61P31/00;A61P35/00;A61P43/00;C07D311/14;C07D335/06;C07D405/12;C07D409/12 主分类号 A61K31/37
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