发明名称 |
COUMARIN DERIVATIVES, METHODS OF PREPARATION AND APPLICATION AS MEDICINES |
摘要 |
The invention concerns compounds of general formula (I) in which: X, X' and X'' independently of each other represent O or S; Y represents O, S, NH or NHS; R3 represents in particular a cycloalkyl group; R5, R6, R7 and R8 mutually identical or different, represent in particular hydrogen; a halogen atom. Said compounds can be used as active substances of medicines as inhibitors of protease. |
申请公布号 |
WO9855472(A1) |
申请公布日期 |
1998.12.10 |
申请号 |
WO1998FR01087 |
申请日期 |
1998.05.29 |
申请人 |
CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE;REBOUD-RAVAUX, MICHELE;POCHET, LIONEL;DOUCET, CAROLINE;PIROTTE, BERNARD;BOGGETTO, NICOLE;DELARGE, JACQUES |
发明人 |
REBOUD-RAVAUX, MICHELE;POCHET, LIONEL;DOUCET, CAROLINE;PIROTTE, BERNARD;BOGGETTO, NICOLE;DELARGE, JACQUES |
分类号 |
A61K31/37;A61K31/4433;A61K31/4436;A61K31/453;A61K31/4709;A61K31/4725;A61P1/18;A61P7/02;A61P9/10;A61P11/00;A61P13/12;A61P17/00;A61P19/02;A61P29/00;A61P31/00;A61P35/00;A61P43/00;C07D311/14;C07D335/06;C07D405/12;C07D409/12 |
主分类号 |
A61K31/37 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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