发明名称 SUBSTITUTED PYRAZOLES AS p38 KINASE INHIBITORS
摘要 A class of pyrazole derivatives is described for use in treating p38 kinase mediated disorders. Compounds of particular interest are defined by Formula (I) wherein R<1>, R<2>, R<3> and R<4> are as described in the specification.
申请公布号 WO9852940(A1) 申请公布日期 1998.11.26
申请号 WO1998US10436 申请日期 1998.05.22
申请人 G.D. SEARLE AND CO.;ANANTANARAYAN, ASHOK;CLARE, MICHAEL;COLLINS, PAUL, W.;CRICH, JOYCE, ZUOWU;DEVRAJ, RAJESH;FLYNN, DANIEL, L.;GENG, LIFENG;HANSON, GUNNAR, J.;KOSZYK, FRANCIS, J.;LIAO, SHUYUAN;PARTIS, RICHARD, A.;RAO, SHASHIDHAR, N.;SELNESS, SHAUN, RAJ;SOUTH, MICHAEL, S.;STEALEY, MICHAEL, A.;WEIER, RICHARD, M.;XU, XIANGDONG 发明人 ANANTANARAYAN, ASHOK;CLARE, MICHAEL;COLLINS, PAUL, W.;CRICH, JOYCE, ZUOWU;DEVRAJ, RAJESH;FLYNN, DANIEL, L.;GENG, LIFENG;HANSON, GUNNAR, J.;KOSZYK, FRANCIS, J.;LIAO, SHUYUAN;PARTIS, RICHARD, A.;RAO, SHASHIDHAR, N.;SELNESS, SHAUN, RAJ;SOUTH, MICHAEL, S.;STEALEY, MICHAEL, A.;WEIER, RICHARD, M.;XU, XIANGDONG
分类号 C07D473/00;A61K31/4155;A61K31/422;A61K31/427;A61K31/4439;A61K31/454;A61K31/4545;A61K31/496;A61K31/498;A61K31/506;A61K31/52;A61K31/5377;A61P1/04;A61P3/14;A61P7/02;A61P9/10;A61P11/00;A61P11/06;A61P17/06;A61P19/02;A61P19/06;A61P29/00;A61P37/06;A61P43/00;C07D401/04;C07D401/14;C07D403/04;C07D405/14;C07D409/04;C07D409/14;C07D413/04;C07D413/14;C07D417/04;C07D417/14;C07D451/02;C07D453/02;C07D471/04 主分类号 C07D473/00
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