发明名称 |
2-heteroaryl-5,11-dihydro-6H-dipyrido[3,2-B:2',3'-E][1,4]diazepines and their use in the prevention or treatment of HIV infection |
摘要 |
PCT No. PCT/US95/01993 Sec. 371 Date Aug. 1, 1996 Sec. 102(e) Date Aug. 1, 1996 PCT Filed Feb. 17, 1995 PCT Pub. No. WO95/22545 PCT Pub. Date Aug. 24, 1995Novel compounds for the treatment of HIV-1 infection. These are 2-heteroary-5,11-dihydro-6H-dipyrido[3,2-b:2',3'-e][1,4]diazepines of the formula=NOR10 and Ar is a group of the formula I, II, III, IV or V <IMAGE> I <IMAGE> II <IMAGE> III <IMAGE> IV <IMAGE> V
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申请公布号 |
US5837704(A) |
申请公布日期 |
1998.11.17 |
申请号 |
US19960663162 |
申请日期 |
1996.08.01 |
申请人 |
BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. |
发明人 |
HARGRAVE, KARL;PROUDFOOT, JOHN;PATEL, USHA;KAPADIA, SURESH;KELLY, TERENCE;MCNEIL, DANIEL;CARDOZO, MARIO |
分类号 |
C07D471/14;(IPC1-7):A61K31/55;A61K243/10;A61K487/12;A61K513/00 |
主分类号 |
C07D471/14 |
代理机构 |
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