发明名称 |
SPIRO-AZACYCLIC DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS |
摘要 |
Substituted spiro-azacyclic derivatives of structural formula (I) are tachykinin receptor antagonists of use, for example, in the treatment or prevention of pain, inflammation, migraine, emesis and postherpetic neuralgia.
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申请公布号 |
CA2287436(A1) |
申请公布日期 |
1998.11.05 |
申请号 |
CA19982287436 |
申请日期 |
1998.04.22 |
申请人 |
MERCK SHARP & DOHME LIMITED |
发明人 |
CURTIS, NEIL ROY;KULAGOWSKI, JANUSZ JOZEF;JACKSON, PHILIP STEPHEN;HOLLINGWORTH, GREGORY JOHN;ELLIOTT, JASON MATTHEW;SWAIN, CHRISTOPHER JOHN;WILLIAMS, BRIAN JOHN;SEWARD, EILEEN MARY |
分类号 |
A61P25/04;A61K31/4192;A61K31/4196;A61K31/427;A61K31/433;A61K31/438;A61K31/4427;A61K31/497;A61K31/501;A61K31/506;A61K31/53;A61P1/08;A61P25/06;A61P29/00;A61P43/00;C07D491/10;C07D491/107;(IPC1-7):C07D491/10;A61K31/445 |
主分类号 |
A61P25/04 |
代理机构 |
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代理人 |
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地址 |
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