发明名称 |
Heterosikl-kondanse morfinoid türevleri(II). |
摘要 |
Formül (I)'in ikameli mono heterosikl-kondanse morfinoid türevleri güçlü ve seçici delta opioid agonist ve antagonistleri olup, analjezik olarak ve normalde delta opioid agonist ve antagonistleri ile tedavi edilebilen patolojik durumlarin tedavisinde kullanilirlar. N=0 veya 1 olup, X,Y,R1-R8 basvuruda tanimlandigi gibidir. |
申请公布号 |
TR9801348(T2) |
申请公布日期 |
1998.10.21 |
申请号 |
TR19980001348T |
申请日期 |
1997.01.08 |
申请人 |
SMITHKLINE BEECHAM S.P.A. |
发明人 |
GIULIO DONDIO;SILVANO RONZONI;PIER ANDREA GATTI;DAVIDE GRAZIANI |
分类号 |
C07F7/18;A61K31/00;A61K31/435;A61K31/439;A61K31/485;A61K31/495;A61K31/496;A61K31/535;A61K31/5375;A61K31/5377;A61P1/00;A61P1/04;A61P1/12;A61P9/00;A61P11/00;A61P11/14;A61P25/08;A61P25/18;A61P25/30;A61P29/00;A61P37/00;A61P37/06;A61P37/08;A61P43/00;C07D471/08;C07D471/10;C07D489/09;C07D491/18;C07D491/20;C07D495/22;C07F7/08;C08G77/12;C08G77/20;C08G77/22;C08G77/50;C08K5/5419;C08L83/04;H05K3/28;(IPC1-7):C07D491/12;C07D495/18;A61K31/445;C07D487/08 |
主分类号 |
C07F7/18 |
代理机构 |
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代理人 |
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地址 |
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