发明名称 PROCESSES AND INTERMEDIATES FOR PREPARING 3-(1-PIPERAZINYL)-1,2-BENZISOTHIAZOLE.
摘要 The present invention relates to processes for the preparation of 3-(1-piperazinyl)-1,2-benzisothiazole or its pharmaceutically acceptable salt and to novel intermediates used in the process. 3-(1-piperazinyl)-1,2-benzisothiazole is a key intermediate useful for the preparation of ziprasidone.
申请公布号 MX9803599(A) 申请公布日期 1998.09.30
申请号 MX19980003599 申请日期 1998.05.06
申请人 PFIZER INCORPORATED 发明人 DARRELL E. FOX;JOHN F. LAMBERT;TERRY G. SINAY JR.;STANLEY W. WALINSKY
分类号 C07D295/22;C07C313/16;C07D275/04;C07D295/26;C07D417/04;(IPC1-7):C07D275/04 主分类号 C07D295/22
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