发明名称 Endothelin-Rezeptor-Antagonisten
摘要 The invention relates to novel compounds of formula I wherein X represents O or S, R<3> represents COOR<4>, CN, 1H-tetrazol-5-yl or CONHSO2R<5>, and at least one of R<2> or R<2'> means a substituent. Said compounds display endothelin receptor antagonistic properties.
申请公布号 DE19710831(A1) 申请公布日期 1998.09.17
申请号 DE19971010831 申请日期 1997.03.15
申请人 MERCK PATENT GMBH, 64293 DARMSTADT, DE 发明人 DORSCH, DIETER, DR., 64372 OBER-RAMSTADT, DE;MEDERSKI, WERNER, DR., 64390 ERZHAUSEN, DE;SCHMITGES, CLAUS-JOCHEN, DR., 64823 GROS-UMSTADT, DE;ANZALI, SOHEILA, DR., 64342 SEEHEIM-JUGENHEIM, DE;OSWALD, MATHIAS, DR., 64673 ZWINGENBERG, DE;WILM, CLAUDIA, DR., 64367 MUEHLTAL, DE;CHRISTADLER, MARIA, 63322 ROEDERMARK, DE
分类号 C07D271/12;C07D285/14;C07D417/06;C07D417/14;(IPC1-7):C07D285/14;C07D417/04;C07D413/06;A61K31/41 主分类号 C07D271/12
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