发明名称 PHARMACEUTICAL PREPARATION COMPRISING LYOPHILIZED LIPOSOMES ENCAPSULATING AN ACTIVE PRINCIPLE WHICH IS HIGHLY INSOLUBLE IN WATER, AND THE PROCESS FOR PREPARING THE SAID PREPARATION
摘要 Lyophilized composition comprising trehalose and lipid liposomes in which a biologically-active principle has been incorporated, characterized in that the biologically-active principle is highly insoluble in water, the trehalose/lipid weight ratio is </= 1.5, and all of the trehalose was added to the outside of the liposomes already formed before lyophilization.
申请公布号 WO9836736(A1) 申请公布日期 1998.08.27
申请号 WO1998EP00817 申请日期 1998.02.12
申请人 ANGELINI RICERCHE S.P.A. SOCIETA' CONSORTILE;CAVALLO, GIOVANNI;MARCHITTO, LEONARDO 发明人 CAVALLO, GIOVANNI;MARCHITTO, LEONARDO
分类号 A61K9/127;A61K31/4045;A61K31/416;A61K38/00;A61K47/26 主分类号 A61K9/127
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