发明名称 SYNTHESIS OF ACYCLIC NUCLEOSIDE DERIVATIVES
摘要 Methods and novel intermediates for the preparation of acyclic nucleoside derivatives of formula (I) where one of R1 and R2 is an amino acid acyl group and the other of R1 and R2 is a -C(O)C3-C21 saturated or monounsaturated, optionally substituted alkyl and R3 is OH or H; or a pharmaceutically acceptable salt thereof.
申请公布号 CA2277151(A1) 申请公布日期 1998.08.13
申请号 CA19982277151 申请日期 1998.02.06
申请人 MEDIVIR AB 发明人 PATEL, RAMESH R.;CHANG, SOU-JEN;TIEN, JIEN-HEH J.;LUKIN, KIRILL L.;KOLACZKOWSKI, LAWRENCE;BHAGAVATULA, LAKSHMI;RASMUSSEN, MICHAEL;NARAYANAN, BIKSHANDARKOR A.;WAYNE, GREG;LANNOYE, GREG;ZHANG, WEIJIANG;TIAN, ZHENPING;RILEY, DAVID A.;MORTON, HOWARD;GATES, BRADLEY D.;SINGAM, PULLA REDDY;LEANNA, M. ROBERT;HANNICK, STEVEN M.
分类号 C12P7/62;A61K31/52;A61P31/12;A61P31/18;A61P31/22;C07C69/16;C07C309/73;C07D473/18;C07D473/40;(IPC1-7):C07D473/18;C07C69/003;C07C229/24;C07C69/66 主分类号 C12P7/62
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