发明名称 DERIVES DE PYRIDONE, LEUR PREPAPARATION ET LEUR UTILISATION COMME INTERMEDIAIRES DE SYNTHESE
摘要 The invention concerns compounds of formula (I) in which: R is -NO2 or -NHR3, R3 being hydrogen, -COR4 (R4 selected among (C1-C4) alkyl, aryl and aryl (C1-C4) alkyl, -COOR5 (R5 selected among (C1-C4) alkyl and aryl (C1-C4) alkyl), -CONHR6 or SO2R6 (R6 selected among (C1-C5) alkyl, aryl and aryl(C1-C4) alkyl), -SO2NR7R8 (R7 and R8 independently of each other represent hydrogen or (C1-C4) alkyl or form with the nitrogen atom a morpholine group), aryl (C1-C4) alkyl, R1 is a (C1-C4) alkyl group linear or branched, cyclo (C3-C8) alkyl, aryl optionally substituted, aryl (C1-C4) alkyl optionally substituted, heteroaryl, R2 is a hydrogen atom, a (C1-C4) alkyl or arylmethyl group, X is an oxygen or sulphur atom, a -CH2-, -SO2- or -NR1- group and Y is a hydrogen atom or (C1-C6) alkyl. The invention is applicable to synthesis intermediates.
申请公布号 FR2758326(A1) 申请公布日期 1998.07.17
申请号 FR19970000378 申请日期 1997.01.16
申请人 SYNTHELABO 发明人 LASSALLE GILBERT;BELLEVERGUE PATRICE;BOURBIER JEAN CLAUDE;GALTIER DANIEL;MARTIN VALERIE
分类号 A61K31/44;A61K31/4436;C07D213/64;C07D213/69;C07D213/70;C07D213/71;C07D213/73;C07D213/75;C07D213/76;C07D405/12;C07D409/06;(IPC1-7):C07D401/06;C07F5/02 主分类号 A61K31/44
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