| 发明名称 |
Synthesis of (4S, 5R) -2, 4-diphenyl-5-carboxy-oxazoline derivative as taxol side-chain precursor |
| 摘要 |
The present invention provides a process for preparing a (4S,5R)-2,4-diphenyl-5-carboxy-oxazoline derivative, which can serve as a taxol side-chain precursor, from the treatment of a (2R,3S)-alkyl trans-3-phenyl-2,3-epoxypropionate derivative with benzonitrile in the presence of a strong acid.
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| 申请公布号 |
US5773629(A) |
申请公布日期 |
1998.06.30 |
| 申请号 |
US19960663736 |
申请日期 |
1996.06.14 |
| 申请人 |
INDUSTRIAL TECHNOLOGY RESEARCH INSTITUTE |
发明人 |
YANG, YUH-LIN ALLEN;GAU, AY-HUA |
| 分类号 |
C07D263/16;(IPC1-7):C07D263/16 |
主分类号 |
C07D263/16 |
| 代理机构 |
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