| 摘要 |
Analgesic 1-(2-[3-(1,2,4,5-tetrahydro-3H,3-benzazepinyl)] alkyl)-1,2,3,4-tetrahydro-4-quinazolinones, 2-(2-[3-(1,2,4,5-tetrahydro-3H,3-benzazepinyl)] alkylamino)benzamides and precursers therefor. Methods are disclosed for preparation of the named compounds. Data regarding symptomatology, analgesic activity, local anesthesia and narcotic antagonism are given. Representative compounds are 1-(2-[3-(1,2,4,5-tetrahydro-3H,3-benzazepinyl)] ethyl) -2-phenyl-1,2,3,4-tetrahydro-4-quinazolinone and 2-(2-[3-(1,2,4,5-tetrahydro-3H,3-benzazepinyl)]ethylamino)benzamide.
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