发明名称 |
BENZAMIDE DERIVATIVES HAVING A VASOPRESSIN ANTAGONISTIC ACTIVITY |
摘要 |
This invention relates to new benzamide derivatives having a vasopressin antagonistic activity, etc. and represented by general formula (I) wherein R<1> is aryl optionally substituted with lower alkoxy, etc., R<2> is lower alkyl, etc., R<3> is hydrogen etc., A is NH, etc., E is (a), etc., X is -CH=CH-, -CH=N-, or S, and Y is a condensed heterocyclic group, etc., and pharmaceutically acceptable salts thereof, to processes for preparation thereof and to a pharmaceutical composition comprising the same. |
申请公布号 |
WO9824771(A1) |
申请公布日期 |
1998.06.11 |
申请号 |
WO1997JP04192 |
申请日期 |
1997.11.18 |
申请人 |
FUJISAWA PHARMACEUTICAL CO., LTD.;SETOI, HIROYUKI;OHKAWA, TAKEHIKO;ZENKOH, TATSUYA;SAWADA, HITOSHI;SAWADA, YUKI;OKU, TERUO |
发明人 |
SETOI, HIROYUKI;OHKAWA, TAKEHIKO;ZENKOH, TATSUYA;SAWADA, HITOSHI;SAWADA, YUKI;OKU, TERUO |
分类号 |
A61K31/40;A61K31/4035;A61K31/41;A61K31/415;A61K31/4184;A61K31/422;A61K31/454;A61K31/495;A61K31/496;A61K31/498;A61K31/517;A61K31/52;A61K31/535;A61K31/5375;A61K31/5377;A61P1/08;A61P1/16;A61P3/10;A61P7/00;A61P9/00;A61P9/12;A61P13/12;A61P43/00;C07C237/42;C07C237/44;C07D209/08;C07D209/12;C07D209/14;C07D209/34;C07D209/42;C07D209/48;C07D215/48;C07D231/56;C07D235/06;C07D235/08;C07D235/10;C07D235/12;C07D235/14;C07D235/16;C07D235/24;C07D235/26;C07D235/28;C07D235/30;C07D235/32;C07D239/88;C07D239/96;C07D241/42;C07D249/18;C07D263/10;C07D263/30;C07D263/54;C07D263/56;C07D265/32;C07D265/34;C07D295/12;C07D295/135;C07D295/18;C07D295/185;C07D401/04;C07D401/06;C07D401/12;C07D403/04;C07D403/06;C07D403/12;C07D413/12;C07D471/04;C07D473/00;C07D487/04;C07D521/00;C07F7/18 |
主分类号 |
A61K31/40 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|