发明名称 METALLOPROTEINASE INHIBITORS
摘要 Compound of formula (I) wherein Ar represents an optionally substituted phenyl or heteroaryl group, m is 1 or 2, n is 0, 1, 2, 3 or 4, X represents -COOH or -CONHOH and R1, R3 and Y are as defined in the specification, are inhibitors of metalloproteinases involved in tissue degradation.
申请公布号 WO9824759(A1) 申请公布日期 1998.06.11
申请号 WO1997GB03316 申请日期 1997.12.02
申请人 BRITISH BIOTECH PHARMACEUTICALS LIMITED;WHITTAKER, MARK;BECKETT, RAYMOND, PAUL;SPAVOLD, ZOE, MARIE;MARTIN, FIONNA, MITCHELL 发明人 WHITTAKER, MARK;BECKETT, RAYMOND, PAUL;SPAVOLD, ZOE, MARIE;MARTIN, FIONNA, MITCHELL
分类号 A61K31/197;A61K31/16;A61K31/164;A61K31/417;A61K31/4402;A61K31/5375;A61P29/00;A61P35/00;A61P43/00;C07C237/22;C07C259/06;C07D213/75;C07D233/24;C07D233/54;C07D233/64;C07D295/12;C07D409/12;(IPC1-7):C07C259/06;C07D295/13;C07C233/51;A61K33/44;A61K31/535;A61K31/415 主分类号 A61K31/197
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