| 发明名称 |
Combinatorial process for synthesizing azetidinone analogs |
| 摘要 |
This invention relates to a combinatorial process for synthesizing a library of azetidinone peptide-like compounds. The compounds are synthesized as mixtures from a common azetidinone intermediate. The compounds are biologically active as inhibitors of the Vasopressin (V1a) receptor.
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| 申请公布号 |
US5759865(A) |
申请公布日期 |
1998.06.02 |
| 申请号 |
US19950433115 |
申请日期 |
1995.05.03 |
| 申请人 |
ELI LILLY AND COMPANY |
发明人 |
BRUNS, ROBERT F.;CHANEY, MICHAEL O.;COOPER, ROBIN D.;HUNDEN, DAVID C.;KOPPEL, GARY A.;SKELTON, JEFFREY J. |
| 分类号 |
C07B61/00;C07D205/085;C07K1/04;C07K5/083;(IPC1-7):G01N33/543;A61K38/00 |
主分类号 |
C07B61/00 |
| 代理机构 |
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