发明名称 PROCESS FOR PREPARATION OF N-DEMETHYL-4-DEOXY-ERYTHROMYCINS A AND B
摘要 A process for the preparation of N-demethyl-4"-deoxy-erythromycins A and B, having formula (I), wherein R<a> is H or OH, by stepwise addition of iodine and base to the N-dimethyl-4"-deoxy-erythromycin, preferably, accompanied by sparging with an inert gas.
申请公布号 WO9822488(A1) 申请公布日期 1998.05.28
申请号 WO1997US20836 申请日期 1997.11.17
申请人 ABBOTT LABORATORIES 发明人 PREMCHANDRAN, RAMIYA, H.;THOMAS, ALBERT, V.;BUSSE, JULIETTE, K.;DETE, JOHN, E.
分类号 C07H17/08;(IPC1-7):C07H17/08 主分类号 C07H17/08
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