摘要 |
Disclosed are novel 2-aryl-5,11-dihydro-6H-dipyrido[3,2-b:2',3'-e][1,4]diazepines. These are useful in the of HIV infection. Exemplary compounds are: 8-Ethyl-1-methyl-10-(4-pyrazolyl)imidazo[2',3':6,5]dipyrido[3,2-b:2',3'-e][1,4]diazepine; 8-c-Propyl-1-methyl-10-(4-pyrazolyl)imidazo[2',3':6,5]dipyrido[3,2-b:2',3'-e][1,4]diazepine; 8-Ethyl-12-methyl-10-(4-pyrazolyl)imidazo[2',3':6,5]dipyrido[3,2-b:2',3'-e][1,4]diazepine; and, 8-c-Propyl-12-methyl-10-(4-pyrazolyl)imidazo[2',3':6,5]dipyrido[3,2-b:2',3 '-e][1,4]diazepine.
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