发明名称 3-ALKOXYCARBONYL-1,3,4-THIADIAZIN-2-ON DERIVATIVES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME
摘要 3-Alkoxycarbonyl-5-heterocyclyl-1,3,4-thiadiazin-2-ones of formula (I) and their salts are new: R<1>-R<3> = H or A; A = 1-6C alkyl; R<4> = 1-15C acyl; R<5> = NH2, NHA, NA2 or satd. 3-8 membered heterocycle contg. 1 or more N atoms (opt. substd. by A) and opt. also contg. NH, NA, O or S in place of 1 CH2 gp.; Q = 1-10C alkylene or a bond; n = 1-3.
申请公布号 HU9600061(A3) 申请公布日期 1998.04.28
申请号 HU19960000061 申请日期 1996.01.10
申请人 MERCK PATENT GMBH., DARMSTADT 发明人
分类号 A61K31/54;A61K31/549;A61K31/55;A61P9/00;A61P9/06;A61P9/08;A61P9/10;A61P43/00;C07D417/04;C07D417/14 主分类号 A61K31/54
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