| 摘要 |
1-(Benzyl or heterocyclylmethyl)-3-(substituted (hetero)aromatic)-fused pyrazole compounds of formula (I) are new. X = O, S NH or CH=CH, and the X-containing ring is optionally substituted by R14; R1 = phenyl, 2-thienyl, 2-pyrrolyl or 2-furanyl, all substituted by R4; R4 = CHOHCH3, 2-6C alkyl (substituted by OH or 1-4C alkoxy), CHO, 1-6C acyl, NO2, 1-6C alkyl (optionally substituted by NH2, N3 or OR5), CH2OR13, or a group of formula (a) or (b); A = phenyl (optionally mono-, di- or trisubstituted by alkyl, alkoxy, alkoxycarbonyl, (each with up to 6C), COOH, NO2, CN, CF3, N3 or halo; R5 = 1-5C acyl, SiR6R7R8, CH2OR10 or a group of formula (c); R6-R8 = 6-10C aryl, 1-6C alkyl; R9, R13 = H or 1-3C alkyl; R10-R12 = H or 1-4C alkyl; R14 = OH, halo, 1-4C alkoxy or 1-4C alkyl; a = 1-3: provided that when R4 = CH2OR13, then A = substituted phenyl where the substituents include alkoxycarbonyl, COOH, NO2, CN, CF3 or N3.
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| 申请人 |
BAYER AG, 51373 LEVERKUSEN, DE |
发明人 |
ROBYR, CHANTAL, DR., 45470 MUELHEIM, DE;STRAUB, ALEXANDER, DR., 42113 WUPPERTAL, DE;JAETSCH, THOMAS, DR., 50668 KOELN, DE;FEURER, ACHIM, DR., 51519 ODENTHAL, DE;KAST, RAIMUND, DR., 42389 WUPPERTAL, DE;STASCH, JOHANNES-PETER, DR., 42651 SOLINGEN, DE;PERZBORN, ELISABETH, DR., 42327 WUPPERTAL, DE;HUETTER, JOACHIM, DR., 42349 WUPPERTAL, DE;DEMBOWSKY, KLAUS, DR., 42115 WUPPERTAL, DE |
