发明名称 |
QUINOLONE- OR NAPHTHYRIDONECARBOXYLIC ACID DERIVATIVE AND SALT THEREOF, PHARMACEUTICAL COMPOSITION CONTAINING THEM AND THEIR USE |
摘要 |
This invention relates to a novel quinolone- or naphthyridone-carboxylic acid derivative or its salt useful as an antibacterial agent, said derivative has a substituent represented by the following formula at the 7 position: <CHEM> wherein preferably R<3> represents at least one member selected from the group consisting of a hydrogen atom, a halogen atom, a substituted or unsubstituted lower alkyl, lower alkoxy or lower alkylthio group, a nitro group, a cyano group, a protected or unprotected hydroxyl group and a protected or unprotected amino group; R<4> represents a hydrogen atom, a substituted or unsubstituted lower alkyl group, a lower alkylidene group and a group forming a cycloalkane ring together with the carbon atom to which R<4> is bonded; and R<5> represents a hydrogen atom or a substituted or unsubstituted lower alkyl or cycloalkyl group. |
申请公布号 |
HUT77314(A) |
申请公布日期 |
1998.03.30 |
申请号 |
HU19970001734 |
申请日期 |
1995.08.04 |
申请人 |
TOYAMA CHEMICAL CO. LTD. |
发明人 |
HAYASHI,KAZUYA;NARITA,HIROKAZU;TAKAHATA,MASAHIRO;TODO,YOZO;WATANABE,YASUO |
分类号 |
C07D401/04;C07D471/04;C07D498/06;C07F7/22 |
主分类号 |
C07D401/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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