发明名称 |
Substituted 1-phenyl-3-pyrazolecarboxamides active on neurotensin receptors, their preparation and pharmaceutical compositions containing them |
摘要 |
The invention relates to new substituted 1-phenyl-3-pyrazolecarboxamides having a great affinity for human neurotensin receptors, to a process for preparing them and to pharmaceutical compositions containing them as active principles. More particularly, this invention relates to the discovery that the affinity for neurotensin receptors, especially human neurotensin receptors, is increased by substituting the phenyl group of 1-phenyl-3-pyrazolecarboxamide compounds with particular groups.
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申请公布号 |
US5723483(A) |
申请公布日期 |
1998.03.03 |
申请号 |
US19960630761 |
申请日期 |
1996.04.10 |
申请人 |
SANOFI |
发明人 |
LABEEUW, BERNARD;GULLY, DANIELLE;JEANJEAN, FRANCIS;MOLIMARD, JEAN-CHARLES;BOIGEGRAIN, ROBERT |
分类号 |
A61K31/415;A61K31/4155;A61K31/42;A61K31/435;A61K31/439;A61K31/44;A61K31/4427;A61K31/4439;A61K31/445;A61K31/454;A61K31/495;A61K31/496;A61K31/535;A61K31/5377;A61P1/00;A61P25/00;A61P35/00;A61P43/00;C07C61/20;C07C62/34;C07C243/22;C07C255/66;C07C309/45;C07C309/47;C07C311/21;C07D231/12;C07D231/14;C07D231/38;C07D233/62;C07D401/10;C07D401/12;C07D403/10;C07D403/12;C07D413/04;C07D413/12;C07D453/02;(IPC1-7):A61K31/415;A01N43/56 |
主分类号 |
A61K31/415 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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