发明名称 |
PROCESS FOR THE PREPARATION OF N-[(1-NBUTYL-4-PIPERIDYL)METHYL] -3,4-DIHYDRO -2H-[1,3] OXAZINO[3,2-A] INDOLE-10-CARBOXAMIDE AND SALTS AND INTERMEDIATES IN THE PROCESS |
摘要 |
<p>A process for the preparation of SB 207266 or a pharmaceutically acceptable salt thereof, which process comprises the reaction of N-(1-nbutyl-4-piperidyl)methylamine with a compound of formula (A), wherein R is alkyl.</p> |
申请公布号 |
CA2263480(A1) |
申请公布日期 |
1998.02.26 |
申请号 |
CA19972263480 |
申请日期 |
1997.08.11 |
申请人 |
SMITHKLINE BEECHAM P.L.C. |
发明人 |
FEDOULOFF, MICHAEL;SMITH, GILLIAN ELIZABETH;STRACHAN, JOHN BRYCE;GUEST, DAVID WILLIAM |
分类号 |
C07D209/42;C07D498/04;(IPC1-7):C07D498/04 |
主分类号 |
C07D209/42 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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