发明名称 |
Oxazolidinone antibacterial agents having a six-membrane heteroaromatic ring |
摘要 |
This invention provides a novel oxazolidinone derivative represented by Formula I or pharmaceutical acceptable salts thereof: <IMAGE> I wherein R1 is substituted or unsubstituted 2-pyrimidinyl, 4-pyrimidinyl, or 3-pyridazinyl; X is hydrogen or fluoro; R3 is C1-4 alkyl, C1-4 alkoxy, C3-6 cycloalkyl or C1-4 alkylamino or dialkylamino. The compounds are useful antimicrobial agents.
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申请公布号 |
US5719154(A) |
申请公布日期 |
1998.02.17 |
申请号 |
US19960762478 |
申请日期 |
1996.12.09 |
申请人 |
TUCKER, JOHN A.;BRICKNER, STEVEN J.;ULANOWICZ, DEBRA A. |
发明人 |
TUCKER, JOHN A.;BRICKNER, STEVEN J.;ULANOWICZ, DEBRA A. |
分类号 |
A61K31/00;A61K31/50;A61K31/501;A61K31/505;A61K31/506;A61P31/00;C07D413/12;(IPC1-7):C07D403/04 |
主分类号 |
A61K31/00 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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