| 发明名称 |
OXYGENATED-HETEROCYCLE CONTAINING SULFONAMIDE INHIBITORS OF ASPARTYL PROTEASE. |
| 摘要 |
<p>The present invention relates to a novel class of sulfonamides which are aspartyl protease inhibitors. This invention also relates to pharmaceutical compositions comprising these compounds. The compounds and pharmaceutical compositions of this invention are particularly well suited for inhibiting HIV-1 and HIV-2 protease activity and consequently, may be advantageously used as anti-viral agents against the HIV-1 and HIV-2 viruses. This invention also relates to methods for inhibiting the activity of HIV aspartyl protease using the compounds of this invention.</p> |
| 申请公布号 |
MX9708055(A) |
申请公布日期 |
1998.01.31 |
| 申请号 |
MX19970008055 |
申请日期 |
1996.04.18 |
| 申请人 |
VERTEX PHARMACEUTICA INCORPORATED |
发明人 |
ROGER D. TUNG;GIVINDA RAO BHISETTI |
| 分类号 |
(IPC1-7):C07D317/24;C07D493/04;C07D307/20;C07D309/12 |
主分类号 |
(IPC1-7):C07D317/24 |
| 代理机构 |
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