发明名称 |
COMPOUNDS FOR AND METHOD OF INHIBITING PHOSPHODIESTERASE IV. |
摘要 |
<p>Novel compounds which are effective PDE IV inhibitors are disclosed. The compounds possess similar or improved PDE IV inhibition as compared to rolipram, with improved selectivity with regard to, e.g., PDE III inhibition. Preferred compounds are 3-(3-cyclopentyloxy-4-methoxy-benzylamino)-4-hydroxymethyl pyrazole and 3-(3-cyclopentyloxy-4-methoxybenzylamino)-4-methoxymethylpyr azole.</p> |
申请公布号 |
MX9700068(A) |
申请公布日期 |
1997.12.31 |
申请号 |
MX19970000068 |
申请日期 |
1995.06.23 |
申请人 |
EURO-CELTIQUE, S.A. |
发明人 |
DAVID CAVALLA;MARK CHASIN;LLOYD DOLBY;RICHARD W. FRITH |
分类号 |
A61K31/41;A61K31/415;A61K31/4164;A61K31/4166;A61K31/42;A61K31/421;A61K31/4245;A61K31/433;A61P11/00;A61P11/06;A61P29/00;A61P37/08;A61P43/00;C07C45/30;C07C235/38;C07C271/00;C07D213/73;C07D213/74;C07D231/12;C07D231/14;C07D231/20;C07D231/38;C07D233/20;C07D233/54;C07D233/64;C07D233/72;C07D233/78;C07D233/88;C07D233/90;C07D239/54;C07D249/04;C07D249/08;C07D249/14;C07D263/34;C07D271/02;C07D275/02;C07D277/10;C07D277/20;C07D277/22;C07D277/24;C07D277/26;C07D277/34;C07D277/38;C07D277/42;C07D285/04;(IPC1-7):C07D231/10;C07D249/00 |
主分类号 |
A61K31/41 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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