发明名称 THROMBIN INHIBITORS
摘要 The present invention provides a compound of general formula (I) in which Y is a primary or secondary amino group; R2 is the residue of a natural or synthetic amino acid; R3 is hydrogen or a C1-C8 alkyl chain which may be substituted by hydroxy or halogen; and X is (CH2)n where n is 1, 2, or 3, or is CH2N or represents a fused phenyl ring which is optionally substituted by one or two methoxy groups or a salt thereof.
申请公布号 WO9746553(A1) 申请公布日期 1997.12.11
申请号 WO1997GB01385 申请日期 1997.05.21
申请人 NOVARTIS AG;BRUNDISH, DEREK, EDWARD;BROWN, LYNDON, NIGEL;LE GRAND, DARREN, MARK;MENEAR, KEITH, ALLAN;SMITH, GARRICK, PAUL;ALLEN, MARK, CHRISTOPHER;BUTLER, PAUL, IAN;COCKROFT, XIAO-LING;MATTHEWS, IAN, TIMOTHY, WILLIAM;WALKER, CLIVE, VICTOR;WATHEY, WILLIAM, BERNARD 发明人 BRUNDISH, DEREK, EDWARD;BROWN, LYNDON, NIGEL;LE GRAND, DARREN, MARK;MENEAR, KEITH, ALLAN;SMITH, GARRICK, PAUL;ALLEN, MARK, CHRISTOPHER;BUTLER, PAUL, IAN;COCKROFT, XIAO-LING;MATTHEWS, IAN, TIMOTHY, WILLIAM;WALKER, CLIVE, VICTOR;WATHEY, WILLIAM, BERNARD
分类号 C07D213/74;C07D401/12;C07D401/14;C07D405/14;C07D413/14;C07D417/14;(IPC1-7):C07D401/12;C07D213/73;A61K31/44;A61K31/445 主分类号 C07D213/74
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