发明名称 |
AMINOTETRALONE DERIVATIVES AND PROCESS FOR PRODUCING THE SAME |
摘要 |
<p>The present invention pertains to a process for the preparation of Compound (4) through the below-described reaction route: <CHEM> wherein R<1> and R<2> each represents H, halogen, OH or C1-6 alkyl group; X and Y each represents a protected amino group and n stands for 0 to 4. According to the above process, an aminotetralone derivative which is an intermediate useful for an industrial preparation of a camptothecin derivative can be obtained in a convenient manner and in a high yield.</p> |
申请公布号 |
EP0811603(A1) |
申请公布日期 |
1997.12.10 |
申请号 |
EP19960903202 |
申请日期 |
1996.02.21 |
申请人 |
DAIICHI PHARMACEUTICAL CO., LTD.;KABUSHIKI KAISHA YAKULT HONSHA |
发明人 |
KAMIHARA, SHINJI;KANAI, KAZUAKI;NOGUCHI, SHIGERU |
分类号 |
C07C231/12;C07C233/41;C07D405/14;C07D491/22;(IPC1-7):C07C233/15;B01J23/44;B01J27/13 |
主分类号 |
C07C231/12 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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