| 发明名称 |
Process for making HIV protease inhibitors |
| 摘要 |
Intermediates of structural formula <IMAGE> can be made by reacting a primary or secondary amine with glycosidol or an activated derivative thereof. The process and intermediates are useful for synthesizing HIV protease inhibitor compounds.
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| 申请公布号 |
US5693803(A) |
申请公布日期 |
1997.12.02 |
| 申请号 |
US19950474800 |
申请日期 |
1995.06.07 |
| 申请人 |
MERCK & CO., INC. |
发明人 |
ASKIN, DAVID;ROSSEN, KAI;REIDER, PAUL;VARSOLONA, RICHARD J.;VOLANTE, RALPH P.;WELLS, KENNETH M. |
| 分类号 |
A61K31/42;A61K31/423;A61K31/44;A61K31/495;A61K31/496;A61P31/12;A61P37/04;A61P43/00;C07D241/04;C07D263/52;C07D303/36;C07D401/06;C07D405/06;C07D413/06;(IPC1-7):C07D405/06;C07D405/14 |
主分类号 |
A61K31/42 |
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