发明名称 2-AMINOINDANS AS SELECTIVE DOPAMINE D3 LIGANDS.
摘要 <p>Compounds and their pharmaceutically acceptable salts suitable for treating central nervous system disorders associated with the dopamine D3 receptor activity of formula (I) wherein R1 and R2 are independently H, C1-8 alkyl or C1-8 alkylAryl; X is CH2R3 or NHSO2R4; Y is hydrogen, CH2R3, NHSO2R4, CONR1R2, SO2NR1R2, SO2CH3, halogen, OSO2CF3, SCH3 or OCH3; R3 is NHSO2R4, SO2R4, CONR1R2 or Aryl; and R4 is NR1R2, C1-C8 alkyl, Aryl or C1-C8 alkylAryl.</p>
申请公布号 MX9705883(A) 申请公布日期 1997.10.31
申请号 MX19970005883 申请日期 1996.01.16
申请人 PHARMACIA & UPJOHN COMPANY 发明人 ARTHUR G. ROMERO;JEFFREY A. LEIBY
分类号 A61K31/135;A61K31/13;A61K31/165;A61K31/18;A61P25/00;A61P25/16;A61P25/20;A61P25/28;A61P25/30;C07C211/42;C07C215/42;C07C233/11;C07C237/20;C07C237/48;C07C311/03;C07C311/05;C07C311/08;C07C311/10;C07C311/18;C07C311/21;C07C311/46;C07C317/06;C07C317/28;C07C317/44;C07C323/28;C07C323/67;C07D213/71;(IPC1-7):C07C211/42;C07C211/10;C07C307/10 主分类号 A61K31/135
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