| 发明名称 |
PROCESS TO MAKE HIV PROTEASE INHIBITOR FROM 2(S)-4-PICOLYL-2-PIPERAZINE-T-BUTYLCARBOXAMIDE |
| 摘要 |
<p>A process for making a clinically efficacious HIV protease inhibitor eliminates one step in its synthesis, by an alternative convergent synthesis using 2(S)-4-picolyl-2-piperazine-t-butylcarboxamide as an intermediate.</p> |
| 申请公布号 |
HRP960114(A2) |
申请公布日期 |
1997.10.31 |
| 申请号 |
HR1996P000114 |
申请日期 |
1996.03.11 |
| 申请人 |
MERCK & CO. INC. |
发明人 |
DAVID ASKIN;KAN K. ENG;PAUL REIDER;RALPH P. VOLANTE |
| 分类号 |
C07D401/06;(IPC1-7):C07D401/06;A61K31/495 |
主分类号 |
C07D401/06 |
| 代理机构 |
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