发明名称 |
Non-steroid androgen receptor antagonist compounds and methods |
摘要 |
Non-steroidal compounds which are high affinity, high specificity ligand antagonists for the androgen receptor are disclosed. Also disclosed are methods for employing the disclosed compounds for modulating processes mediated by the androgen receptor and for treating patients requiring androgen receptor antagonist therapy.
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申请公布号 |
US5677336(A) |
申请公布日期 |
1997.10.14 |
申请号 |
US19930141492 |
申请日期 |
1993.10.21 |
申请人 |
LIGAND PHARMACEUTICALS INCORPORATED |
发明人 |
JONES, TODD K.;HAMANN, LAWRENCE G.;FARMER, LUC;JOHNSON, MICHAEL G.;GOLDMAN, MARK E. |
分类号 |
A61K31/04;A61K31/05;A61K31/075;A61K31/12;A61K31/22;C07C39/23;C07C43/23;C07C45/67;C07C45/71;C07C47/575;C07C49/753;C07C69/017;C07C205/06;C07C205/18;C07C205/45;(IPC1-7):A61K31/04;A61K31/085 |
主分类号 |
A61K31/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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