发明名称 PARA-SUBSTITUTED PHENYLPROPANOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS
摘要 The present invention relates to a class of compounds represented by Formula (I) or a phramaceutically acceptable salt thereof, pharmaceutical composition comprising compounds of Formula (I), and methods of selectively inhibiting or antagonizing the alpha v beta 3 integrin.
申请公布号 WO9736859(A1) 申请公布日期 1997.10.09
申请号 WO1997US04460 申请日期 1997.03.26
申请人 G.D. SEARLE & CO.;CHEN, BARBARA, B.;CHEN, HELEN, Y.;GESICKI, GLEN, J.;HAACK, RICHARD, A.;MALECHA, JAMES, W.;PENNING, THOMAS, D.;RICO, JOSEPH, G.;ROGERS, THOMAS, E.;RUMINSKI, PETER, G.;RUSSELL, MARK, A.;YU, STELLA, S. 发明人 CHEN, BARBARA, B.;CHEN, HELEN, Y.;GESICKI, GLEN, J.;HAACK, RICHARD, A.;MALECHA, JAMES, W.;PENNING, THOMAS, D.;RICO, JOSEPH, G.;ROGERS, THOMAS, E.;RUMINSKI, PETER, G.;RUSSELL, MARK, A.;YU, STELLA, S.
分类号 A61K31/155;A61K31/166;A61K31/17;A61K31/18;A61K31/216;A61K31/4168;A61K31/4192;A61K31/4453;A61K31/505;A61K31/5375;A61P9/14;A61P19/08;A61P19/10;A61P27/02;A61P35/00;C07C257/18;C07C259/18;C07C275/42;C07C279/18;C07C279/22;C07C279/24;C07C279/28;C07C311/06;C07C311/13;C07C311/19;C07C311/47;C07C311/64;C07C317/44;C07C323/52;C07D223/12;C07D233/50;C07D233/88;C07D239/14;C07D249/14;C07D271/06;C07D271/07;C07D295/20;C07D295/215;C07D521/00;(IPC1-7):C07C279/18;C07D223/04 主分类号 A61K31/155
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