发明名称 Process for the preparation of 1,3-dimethyl-5-fluoro-pyrazole-4-carboxanilides
摘要 A new process for the preparation of a known 1,3-dimethyl-5-fluoro-pyrazole-4-carboxanilide of the formula <IMAGE> in which Ar represents optionally substituted phenyl, which process comprises a) reacting in a first stage, 1,3-dimethyl-5-chloro-pyrazole-4-carbonyl chloride with a fluoride, if appropriate in the presence of a diluent, and b) reacting in a second stage, the 1,3-dimethyl-5-fluoro-pyrazole-4-carbonyl fluoride obtained in this reaction with an aniline of the formulaH2N-Arin which Ar has the abovementioned meaning, if appropriate in the presence of an acid acceptor and if appropriate in the presence of a diluent. 1,3-Dimethyl-5-fluoro-pyrazole-4-carbonyl fluoride as a new compound.
申请公布号 US5675016(A) 申请公布日期 1997.10.07
申请号 US19960755678 申请日期 1996.11.25
申请人 BAYER AKTIENGESELLSCHAFT 发明人 GALLENKAMP, BERND;ROHE, LOTHAR;MARHOLD, ALBRECHT
分类号 C07D231/16;A01N43/56;C07D231/14;(IPC1-7):C07D231/16 主分类号 C07D231/16
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