The present invention provides a method for synthesizing indolylmaleimides by reacting an activated maleimide preferably with an optionally substituted organometallic-3-indole in the presence of a transition metal catalyst.
申请公布号
WO9734890(A1)
申请公布日期
1997.09.25
申请号
WO1997US04416
申请日期
1997.03.20
申请人
ELI LILLY AND COMPANY;FAUL, MARGARET, M.;JIROUSEK, MICHAEL, R.;MCDONALD, JOHN, HAMPTON, III;NEEL, DAVID
发明人
FAUL, MARGARET, M.;JIROUSEK, MICHAEL, R.;MCDONALD, JOHN, HAMPTON, III;NEEL, DAVID