发明名称 |
Novel crystal form of anhydrous 7-(Ä1alpha, 5alpha, 6alphaÜ-6-amino-3-azabicyclo Ä3.1.0Ü hex-3-yl)-6-fluoro-1-(2,4-difluorophenyl)-1,4- dihydro-4-oxo-1,8-naphthyridine-3-carboxylic acid methanesulfonic acid salt |
摘要 |
New crystal form, (I'), of 7-([1~a, 5~a, 6~a]-6-amino-3-azabicyclo [3.1.0] hex-3-yl)-6- fluoro-1-(2,4-difluorophenyl)- 1,4-dihydro-4-oxo-1,8- naphthyridine-3-carboxylic acid, methanesulphonic acid salt (I), is characterised by the following major peaks in its X-ray powder diffraction pattern: Peak number; 2~h( deg )Cu; d space: (1; 4.5; 19.5); (2; 7.7; 11.5); (3; 9.1; 9.7); (4; 13.6; 6.5); (5; 15.0; 5.9); (6; 18.2; 4.9); (7; 18.6; 4.8); (8; 22.8; 3.9). |
申请公布号 |
OA10293(A) |
申请公布日期 |
1997.09.19 |
申请号 |
OA19960060835 |
申请日期 |
1996.06.06 |
申请人 |
PFIZER INC. |
发明人 |
HANDANYAN, LYNNE, A.;HENDRICKSON, ROBERT, L.;JOHNSON, PHILLIP, J.;MORRIS, THOMAS, A.;NORRIS TIMOTHY |
分类号 |
C07D487/04;A61K;A61K31/00;A61K31/395;A61K31/435;A61K31/4375;A61K31/44;A61K31/495;A61P31/04;C07C303/00;C07C309/00;C07C311/00;C07D;C07D221/00;C07D221/04;C07D471/02;C07D471/04;C07D519/00;(IPC1-7):C07D471/04 |
主分类号 |
C07D487/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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