发明名称 |
MCBI ANALOGS OF CC-1065 AND THE DUOCARMYCINS |
摘要 |
MCBI (7-methoxy-1,2,9,9a-tetra-hydrocyclopropa[c]benz[e]indol-4-one) is employable as a DNA alkylating agent and can be incorporated into analogs of CC-1065 and the duocarmycins for constructing regioselective DNA alkylating agents.
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申请公布号 |
WO9732850(A1) |
申请公布日期 |
1997.09.12 |
申请号 |
WO1997US03641 |
申请日期 |
1997.03.07 |
申请人 |
THE SCRIPPS RESEARCH INSTITUTE;BOGER, DALE, L. |
发明人 |
BOGER, DALE, L. |
分类号 |
A61K31/00;A61K31/40;A61K31/403;A61K31/407;A61P35/00;C07D209/60;C07D209/70;C07D209/94;C07D487/04;C07D519/00;(IPC1-7):C07D209/70;C07D403/06;C07D403/14 |
主分类号 |
A61K31/00 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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