发明名称 (THIOPHEN-2-YL)-PIPERIDIN OR TETRAHYDROPYRIDIN CARBOXAMIDES.
摘要 <p>This invention provides compounds having formula (I), wherein R is hydrogen, alkyl, alkenyl, alkynyl, -COR2, phenyl, or phenylalkyl of 7-10 carbon atoms; the dotted line represents an optional double bond; R1 is hydrogen, -OH, OR3, or is absent if the optional double bond is present; R2 and R3 are each, independently, alkyl, alkenyl, alkynyl, phenyl, or phenylalkyl; R4 is hydrogen, -OR5, alkyl, alkenyl, alkynyl, -COR5, -CO2R5, -CONR5R6, perhaloalkyl, halogen, phenyl, or phenylalkyl; R5 and R6 are each, independently, hydrogen, alkyl, alkenyl, alkynyl, phenyl, or phenylalkyl; and n = 0 - 2 or a pharmaceutically acceptable salt thereof that are useful as antipsychotic, antidepressant and anxiolytic agents useful in the treatment and relief of the symptoms of these disease states.</p>
申请公布号 MX9703894(A) 申请公布日期 1997.08.30
申请号 MX19970003894 申请日期 1995.11.22
申请人 AMERICAN HOME PRODUCTS CORPORATION 发明人 REINHARDT BERNHARD BAUDY
分类号 A61K31/4433;A61K31/445;A61K31/55;A61P25/00;A61P25/20;A61P25/24;A61P25/26;A61P43/00;C07D409/04;C07D409/14;(IPC1-7):C07D409/04 主分类号 A61K31/4433
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