N-heterocyclic moiety containing hydroxyethylamine compounds are effective as retroviral protease inhibitors, and in particular as inhibitors of HIV protease.
申请公布号
US5643924(A)
申请公布日期
1997.07.01
申请号
US19950455237
申请日期
1995.05.31
申请人
MONSANTO COMPANY OF ST. LOUIS
发明人
TALLEY, JOHN J.;GETMAN, DANIEL P.;DECRESCENZO, GARY A.;REED, KATHRYN L.;LIN, KO-CHUNG;FRESKOS, JOHN NICHOLAS;CLARE, MICHAEL;ROGIER, JR., DONALD JOSEPH;HEINTZ, ROBERT M.;VAZQUEZ, MICHAEL L.;MUELLER, RICHARD A.