发明名称 DIHYDRATE DU (2R,3S)-3-TERT-BUTOXYCARBONYLAMINO-2-HYDROXY- 3-PHENYLPROPIONATE DE 4,10BETA-DIACETOXY-2ALPHA-BENZOYLOXY- 5BETA,2O-EPOXY-1-HYDROXY-9-OXO-19-NOR-CYCLOPROPA(G)TAX-11- ENE-13ALPHA-YLE, ET SON PROCEDE DE PREPARATION
摘要 A 4,10 beta -diacetoxy-2 alpha -benzoyloxy-5 beta ,20-epoxy-1-hydroxy-9-oxo-19-nor-cyclopropa[g]tax-11-ene-13 alpha -yl (2R,3S)-3-tert-butoxycarbonylamino-2-hydroxy-3-phenylpropionate dihydrate, and the preparation thereof by crystallisation from a water-alcohol or water-ketone solution, are disclosed.
申请公布号 FR2742438(A1) 申请公布日期 1997.06.20
申请号 FR19950014841 申请日期 1995.12.14
申请人 RHONE POULENC RORER SA 发明人 AUTHELIN JEAN RENE;DIDIER ERIC;LAVIGNE MICHEL
分类号 A61K31/335;C07D305/14 主分类号 A61K31/335
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