发明名称 |
DIHYDRATE DU (2R,3S)-3-TERT-BUTOXYCARBONYLAMINO-2-HYDROXY- 3-PHENYLPROPIONATE DE 4,10BETA-DIACETOXY-2ALPHA-BENZOYLOXY- 5BETA,2O-EPOXY-1-HYDROXY-9-OXO-19-NOR-CYCLOPROPA(G)TAX-11- ENE-13ALPHA-YLE, ET SON PROCEDE DE PREPARATION |
摘要 |
A 4,10 beta -diacetoxy-2 alpha -benzoyloxy-5 beta ,20-epoxy-1-hydroxy-9-oxo-19-nor-cyclopropa[g]tax-11-ene-13 alpha -yl (2R,3S)-3-tert-butoxycarbonylamino-2-hydroxy-3-phenylpropionate dihydrate, and the preparation thereof by crystallisation from a water-alcohol or water-ketone solution, are disclosed. |
申请公布号 |
FR2742438(A1) |
申请公布日期 |
1997.06.20 |
申请号 |
FR19950014841 |
申请日期 |
1995.12.14 |
申请人 |
RHONE POULENC RORER SA |
发明人 |
AUTHELIN JEAN RENE;DIDIER ERIC;LAVIGNE MICHEL |
分类号 |
A61K31/335;C07D305/14 |
主分类号 |
A61K31/335 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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