发明名称 SUBSTITUTED PIPERIDINE DERIVATIVES AS SELECTIVE AGONISTS OF 5-HT RECEPTORS
摘要 A compound of formula (I), or a salt or prodrug thereof, wherein G is attached at position 3 or 4 of the piperidine ring and represents halogen or C1-6 alkoxy; R<1> represents C3-6 alkenyl, C3-6 alkynyl, aryl(C1-6)alkyl or heteroaryl(C1-6)alkyl, any of which groups may be optionally substituted; processes for its preparation and its use in therapy, particularly in the treatment of migraine.
申请公布号 WO9718202(A1) 申请公布日期 1997.05.22
申请号 WO1996GB02765 申请日期 1996.11.13
申请人 MERCK SHARP & DOHME LIMITED;CASTRO PINEIRO, JOSE LUIS;COLLINS, IAN, JAMES;MACLEOD, ANGUS, MURRAY;MOYES, CHRISTOPHER, RICHARD;ROWLEY, MICHAEL;SHOWELL, GRAHAM, ANDREW 发明人 CASTRO PINEIRO, JOSE LUIS;COLLINS, IAN, JAMES;MACLEOD, ANGUS, MURRAY;MOYES, CHRISTOPHER, RICHARD;ROWLEY, MICHAEL;SHOWELL, GRAHAM, ANDREW
分类号 C07D521/00;(IPC1-7):C07D401/14;C07D409/14;A61K31/445 主分类号 C07D521/00
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