摘要 |
A compound of formula (I), or a salt or prodrug thereof, wherein G is attached at position 3 or 4 of the piperidine ring and represents halogen or C1-6 alkoxy; R<1> represents C3-6 alkenyl, C3-6 alkynyl, aryl(C1-6)alkyl or heteroaryl(C1-6)alkyl, any of which groups may be optionally substituted; processes for its preparation and its use in therapy, particularly in the treatment of migraine.
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申请人 |
MERCK SHARP & DOHME LIMITED;CASTRO PINEIRO, JOSE LUIS;COLLINS, IAN, JAMES;MACLEOD, ANGUS, MURRAY;MOYES, CHRISTOPHER, RICHARD;ROWLEY, MICHAEL;SHOWELL, GRAHAM, ANDREW |
发明人 |
CASTRO PINEIRO, JOSE LUIS;COLLINS, IAN, JAMES;MACLEOD, ANGUS, MURRAY;MOYES, CHRISTOPHER, RICHARD;ROWLEY, MICHAEL;SHOWELL, GRAHAM, ANDREW |