发明名称 Process for the preparation of ethyl 3S-[[4-[[4-(aminoiminomethyl)phenyl]amino]-1,4-dioxobutyl]amino]-4-pentynoate
摘要 The present invention relates to a novel process for the preparation of ethyl 3S-[[4-[[4-(aminoiminomethyl)phenyl]amino]-1,4-dioxobutyl]amino]-4-pentynoate and pharmaceutically acceptable acid addition salt thereof.
申请公布号 US5631399(A) 申请公布日期 1997.05.20
申请号 US19960647514 申请日期 1996.05.14
申请人 G. D. SEARLE & CO. 发明人 BABIAK, KEVIN A.;BABU, SRINIVASAN;BEHLING, JAMES R.;BOYS, MARK L.;CAIN-JANICKI, KIMBERLY J.;DOUBLEDAY, WENDEL W.;FARID, PAYMAN;HAGEN, TIMOTHY J.;HALLINAN, E. A.;HANSEN, JR., DONALD W.;KORTE, DONALD E.;MC LAUGHLIN, KATHLEEN T.;MEDICH, JOHN R.;NUGENT, SEAN T.;ORLOVSKI, VLASDISLAV;PARK, JUNG M.;PETERSON, KAREN B.;PILIPAUSKAS, DANIEL R.;PITZELE, BARNETT S.;TSYMBALOV, SOFYA;STAHL, GLENN L.
分类号 C07C227/02;C07B61/00;C07C227/12;C07C227/34;C07C229/08;C07C257/18;(IPC1-7):C07C229/30 主分类号 C07C227/02
代理机构 代理人
主权项
地址