| 摘要 |
Peptide derivatives from the group comprising Bit-Gly-Gly-Gly-Arg-Gly-Asp-Ser-Pro-Lys-OH, Bit-Gly-Gly-Gly-Lys-Thr-Ala-Asp-Cys(Trt)-Pro-OH, cyclo-(Arg-Gly-Asp-D-Phe-Lys(N'epsilon'-Bit)), cyclo-(Arg-Gly-Asp-D-Phe-Lys(N'epsilon'-Aha)), cyclo-(Arg-Gly-Asp-D-Phe-Lys(N'epsilon'-Bit-Aha)-Gly), cyclo-(Arg-Gly-Asp-D-Phe-Val-Lys(N'epsilon'-Bit-Aha)), cyclo-(Arg-Gly-Asp-D-Phe-N-Me-Lys(N'epsilon'-Bit-Aha)), cyclo-(Arg-Gly-Asp-D-Phe-Lys(N'epsilon'-Bit-Aha)), cyclo-(Arg-Gly-Asp-D-Phe-Lys(BOC-Aha)) and pharmaceutically acceptable salts thereof, which are as integrin inhibitors usable for production of pharmaceutical compositions and for other purposes in biology and molecular biology. |
