发明名称 CONJUGATES USEFUL IN THE TREATMENT OF BENIGN PROSTATIC HYPERPLASIA
摘要 Novel pharmaceutical compositions useful for the treatment of benign prostatic hyperplasia which comprises novel oligopeptides, which are selectively cleaved by enzymatically active PSA, in conjugation with a cytotoxic agent are described. Methods of treating benign prostate hypertrophy are also disclosed.
申请公布号 WO9714416(A1) 申请公布日期 1997.04.24
申请号 WO1996US16490 申请日期 1996.10.15
申请人 MERCK & CO., INC.;DEFEO-JONES, DEBORAH;JONES, RAYMOND, E.;OLIFF, ALLEN, I.;SCOLNICK, EDWARD, M.;GARSKY, VICTOR, M. 发明人 DEFEO-JONES, DEBORAH;JONES, RAYMOND, E.;OLIFF, ALLEN, I.;SCOLNICK, EDWARD, M.;GARSKY, VICTOR, M.
分类号 C07H15/252;A61K31/00;A61K31/24;A61K31/335;A61K31/337;A61K31/40;A61K31/407;A61K31/475;A61K31/505;A61K31/513;A61K31/517;A61K31/529;A61K31/675;A61K31/70;A61K31/7028;A61K31/7034;A61K31/704;A61K31/7042;A61K31/7048;A61K38/00;A61K45/00;A61K47/42;A61K47/48;A61P13/00;A61P13/08;C07K7/06;C07K7/08;C07K14/47;(IPC1-7):A61K31/40;A61K31/44;A61K38/02;A61K38/07;A61K38/08;A61K38/10;A61K38/14 主分类号 C07H15/252
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