发明名称 CEPHALOSPORIN COMPOUNDS AND PRODUCTION THEREOF
摘要 <p>Cephalosporin compounds represented by general formula (I), pharmacologically acceptable addition salts thereof, method for the production thereof, and medicinal uses thereof, wherein R<1> represents hydrogen or lower alkyl, and R<2> represents 1-alkanoyloxyalkyl or 1-alkoxycarbonyloxy-alkyl. These compounds and salts not only can be readily absorbed through the digestive tract to exhibit wide antibacterial activities in vivo in the form of the hydrolyzates thereof, but also have remarkable sweetness 10 to 400 times as high as that of sucrose. Therefore they are useful in preventing and treating infectious diseases by oral administration. <CHEM></p>
申请公布号 EP0497978(B1) 申请公布日期 1997.04.16
申请号 EP19900915817 申请日期 1990.10.24
申请人 KYOTO PHARMACEUTICAL INDUSTRIES, LTD. 发明人 MURO, HIROYUKI;KASAI, MASAYASU;HATANO, SATORU;NISHIMURA, KEN-ICHI;NISHIZAWA, SUSUMU;KAKEYA, NOBUHARU
分类号 A61K31/545;A61K31/546;A61P31/04;C07D501/00;C07D501/20;C07D501/22;(IPC1-7):C07D501/20 主分类号 A61K31/545
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